SCHEMBL9846194

SCHEMBL9846194

CCc1cc(/C=C/c2cc(CC)c(C)[nH]c2=O)c(OC)nc1C

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 5/20 0.36
PDE3A Q14432 5/20 0.36
HCAR2 Q8TDS4 2/20 0.33
TYMS P04818 1/20 0.32
PDE10A Q9Y233 3/20 0.32
LMNA P02545 2/20 0.31
MEN1 O00255 1/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
KDM4E B2RXH2 1/20 0.30
HSD17B10 Q99714 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846195 1.00 PDE3B (0.36) PDE3BPDE3AHCAR2TYMSPDE10A
SCHEMBL9846206 0.78 PDE3B (0.40) PDE3BPDE3AHCAR2PDE10AALDH1A1
SCHEMBL9680874 0.78 CDK5 (0.39) PDE3BPDE3AHCAR2PDE10AMEN1
SCHEMBL9680870 0.78 CDK5 (0.39) PDE3BPDE3AHCAR2PDE10AMEN1
SCHEMBL11894731 0.75 PDE3B (0.35) PDE3BPDE3AHCAR2
SCHEMBL9267418 0.75 ALDH1A1 (0.39) LMNAALDH1A1KDM4E
SCHEMBL9846217 0.74 PDE3B (0.37) PDE3BPDE3AHCAR2PDE10AALDH1A1
SCHEMBL9333881 0.73 MAPT (0.35) PDE3BPDE3AHCAR2LMNAALDH1A1
SCHEMBL9431796 0.73 ALDH1A1 (0.43) LMNAALDH1A1RAB9AMAPK1
SCHEMBL9431804 0.73 ALDH1A1 (0.43) LMNAALDH1A1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed