SCHEMBL9680967

SCHEMBL9680967

Fc1cccc(F)c1-c1ccno1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.42
RAB9A P51151 4/20 0.42
NPC1 O15118 3/20 0.42
LMNA P02545 1/20 0.42
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
PDE4B Q07343 2/20 0.37
CASP3 P42574 3/20 0.37
SENP8 Q96LD8 3/20 0.37
SENP7 Q9BQF6 3/20 0.37
SENP6 Q9GZR1 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP1A2 P05177 3/20 0.36
CYP19A1 P11511 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
EPHX2 P34913 1/20 0.35
GAA P10253 2/20 0.35
MGAM O43451 1/20 0.35
SI P14410 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24977286 0.86 EPHX2 (0.41) NOTUMRAB9ANPC1LMNAKDM4E
SCHEMBL29541410 0.80 NOTUM (0.41) NOTUMRAB9ANPC1KDM4EALDH1A1
SCHEMBL29541827 0.77 BCAT1 (0.46) NOTUMRAB9ANPC1KDM4EALDH1A1
SCHEMBL7843687 0.76 NOTUM (0.50) NOTUMRAB9ANPC1LMNAKDM4E
SCHEMBL29541546 0.76 CYP1A2 (0.47) NOTUMRAB9ANPC1KDM4EALDH1A1
SCHEMBL6817772 0.76 CYP1A2 (0.47) NOTUMRAB9ANPC1KDM4EALDH1A1
SCHEMBL14125002 0.74 NOTUM (0.56) NOTUMRAB9ANPC1KDM4EALDH1A1
SCHEMBL4053984 0.74 EPHX2 (0.49) NOTUMRAB9AKDM4EALDH1A1CYP1A2
SCHEMBL24978464 0.72 SYK (0.55) RAB9ANPC1CYP1A2CYP19A1CYP2C9
SCHEMBL3689041 0.68 NPC1 (0.35) RAB9ANPC1LMNAPDE4BCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486782-A1 Improved process for the synthesis of alpha-((dialkylamino)substituted-methylene)-beta-oxo-(substituted) propanenitriles AMERICAN CYANAMID COMPANY (US) 1992-05-27 EP claimed
US-5103015-A 5-(substituted)isoxazole compounds AMERICAN CYANAMID COMPANY (US) 1992-04-07 US claimed
US-11306078-B2 Piperidine CXCR7 receptor modulators IDORSIA PHARMACEUTICALS LTD. (CH) 2022-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11306078-B2 Piperidine CXCR7 receptor modulators CXCR1, CXCR5, ACKR3 NOTUM 4727/4885RAB9A 1065/4885NPC1 1403/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.