SCHEMBL6817772

SCHEMBL6817772

Fc1ccccc1-c1ccno1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP19A1 P11511 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
KMT2A Q03164 3/20 0.42
PKM P14618 2/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
MEN1 O00255 2/20 0.42
NFKB1 P19838 1/20 0.42
MAPK1 P28482 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
EPHX2 P34913 1/20 0.42
NOTUM Q6P988 3/20 0.41
ADRA1A P35348 3/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1B P35368 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29541546 1.00 CYP1A2 (0.47) CYP1A2CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL29541827 0.83 BCAT1 (0.46) CYP1A2CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL4053984 0.80 EPHX2 (0.49) CYP1A2CYP19A1CYP2C9CYP2C19RAB9A
SCHEMBL3609355 0.80 NPC1 (0.50) NPC1RAB9AKMT2APKMSMN1; SMN2
SCHEMBL2415309 0.77 EPHX2 (0.58) CYP1A2CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL6368033 0.77 ALDH1A1 (0.48) CYP1A2CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL12681544 0.77 SMN1; SMN2 (0.51) CYP1A2CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL7450169 0.77 CYP1A2 (0.46) CYP1A2CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL29503805 0.77 SMN1; SMN2 (0.51) CYP1A2CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL2310167 0.77 CYP1A2 (0.46) CYP1A2CYP19A1CYP2C9CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486782-A1 Improved process for the synthesis of alpha-((dialkylamino)substituted-methylene)-beta-oxo-(substituted) propanenitriles AMERICAN CYANAMID COMPANY (US) 1992-05-27 EP claimed
US-5103015-A 5-(substituted)isoxazole compounds AMERICAN CYANAMID COMPANY (US) 1992-04-07 US claimed
US-20230024012-A1 Protease Inhibitors for Treatment of Coronavirus Infections THE SCRIPPS RESEARCH INSTITUTE 2023-01-26 US disclosed
US-20040110802-A1 Antibacterial benzoic acid derivatives PHARMACIA & UPJOHN COMPANY 2004-06-10 US disclosed
WO-2004018428-A1 ANTIBACTERIAL BENZOIC ACID DERIVATIVES PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230024012-A1 Protease Inhibitors for Treatment of Coronavirus Infections ACE, ACE2, TMPRSS2 CYP1A2 318/4885CYP19A1 1015/4885CYP2C9 277/4885
US-20040110802-A1 Antibacterial benzoic acid derivatives GABRD, GABBR1, GABRA1 CYP1A2 710/4885CYP19A1 869/4885CYP2C9 903/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.