SCHEMBL9681202

SCHEMBL9681202

Fc1ccc2c(N3CCNCC3)nn(-c3ccccc3F)c2c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.44
SCN5A Q14524 2/20 0.44
SCN2A Q99250 1/20 0.44
SCN3A Q9NY46 1/20 0.44
SCN8A Q9UQD0 1/20 0.44
HTR1A P08908 4/20 0.43
SLC6A2 P23975 3/20 0.43
SLC6A4 P31645 3/20 0.43
HTR7 P34969 1/20 0.42
KHK P50053 4/20 0.41
SLC6A3 Q01959 1/20 0.40
MAPT P10636 1/20 0.39
HTR3A P46098 1/20 0.39
HTR6 P50406 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9682493 0.88 ADRB1 (0.50) HTR1ASLC6A2SLC6A4HTR7KHK
SCHEMBL9683176 0.87 SCN9A (0.48) SCN9ASCN5ASCN2ASCN3ASCN8A
Hydrochloric Acid SCHEMBL9681905 0.86 SCN9A (0.47) SCN9ASCN5ASCN2ASCN3ASCN8A
SCHEMBL9683217 0.85 SCN9A (0.42) SCN9ASCN5ASCN2ASCN3ASCN8A
SCHEMBL9681244 0.85 KHK (0.57) KHKHTR3A
SCHEMBL9683240 0.82 KHK (0.50) HTR1AHTR7KHKHTR6
SCHEMBL8128906 0.77 HRH4 (0.44) HTR1ASLC6A2SLC6A4HTR7KHK
SCHEMBL9682532 0.75 KHK (0.51) HTR1ASLC6A2HTR7KHKSLC6A3
SCHEMBL9681305 0.74 KHK (0.47) HTR1ASLC6A2SLC6A4HTR7KHK
SCHEMBL9682462 0.74 KHK (0.44) HTR1ASLC6A2SLC6A4HTR7KHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed