SCHEMBL9681273

SCHEMBL9681273

Clc1ccc2c(N3CCNCC3)nn(-c3ccccc3)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 13/20 0.57
HTR3E A5X5Y0 1/20 0.48
HTR3B O95264 1/20 0.48
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
ADRB1 P08588 1/20 0.48
CYP3A4 P08684 1/20 0.48
HTR1A P08908 1/20 0.48
CYP2D6 P10635 1/20 0.48
THRB P10828 1/20 0.48
CYP2C9 P11712 1/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
SLC6A4 P31645 1/20 0.48
CYP2C19 P33261 1/20 0.48
HTR7 P34969 1/20 0.48
HTR2B P41595 1/20 0.48
HTT P42858 1/20 0.48
HTR3A P46098 1/20 0.48
HTR6 P50406 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9681879 0.99 KHK (0.56) KHKHTR3EHTR3BTP53CYP1A2
SCHEMBL9680691 0.85 KHK (0.57) KHKHTR3EHTR3BADRB1HTT
SCHEMBL9681923 0.85 MAT2A (0.65) KHKTP53HTR6MAT2AKDM4E
SCHEMBL9681244 0.85 KHK (0.57) KHKHTR3EHTR3BADRB1HTR3A
SCHEMBL2710715 0.84 KHK (0.54) KHKHTR3EHTR3BADRB1HTR2C
Hydrochloric Acid SCHEMBL9681346 0.82 KHK (0.53) KHKHTR3EHTR3BADRB1HTR2C
SCHEMBL10582090 0.81 MAT2A (0.47) KHKMAT2ANPSR1
Fumaric Acid SCHEMBL9681264 0.77 MAT2A (0.59) KHKTP53HTR2AHTTMAT2A
Fumaric Acid SCHEMBL9681259 0.77 MAT2A (0.59) KHKTP53HTR2AHTTMAT2A
SCHEMBL9682532 0.77 KHK (0.51) KHKHTR3EHTR3BCYP1A2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed