SCHEMBL9682530

SCHEMBL9682530

CN1CCN(c2nn(-c3ccc(F)cc3)c3cc(F)ccc23)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 3/20 0.51
HTR3E A5X5Y0 2/20 0.43
HTR3B O95264 2/20 0.43
HTR3A P46098 2/20 0.43
HTR3D Q70Z44 2/20 0.43
HTR3C Q8WXA8 2/20 0.43
LMNA P02545 2/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
HRH4 Q9H3N8 4/20 0.41
TRPV4 Q9HBA0 1/20 0.40
TNKS O95271 1/20 0.40
PARP1 P09874 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680590 0.92 KHK (0.58) KHKHTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL9682507 0.91 KHK (0.57) KHKHTR3EHTR3BHTR3AHTR3D
SCHEMBL9681940 0.86 KHK (0.48) KHKHTR3EHTR3BHTR3AHTR3D
SCHEMBL9683240 0.84 KHK (0.50) KHKHRH4HTR6
Fumaric Acid SCHEMBL9681236 0.78 LMNA (0.44) KHKLMNANPC1TP53RAB9A
Fumaric Acid SCHEMBL9681228 0.78 LMNA (0.44) KHKLMNANPC1TP53RAB9A
SCHEMBL9681923 0.76 MAT2A (0.65) KHKNPC1TP53RAB9AALDH1A1
SCHEMBL9681244 0.76 KHK (0.57) KHKHTR3EHTR3BHTR3AHTR3D
SCHEMBL6125292 0.74 KHK (0.56) KHKHTR3EHTR3BHTR3AHTR3D
SCHEMBL9683181 0.74 KHK (0.57) KHKHTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed