SCHEMBL9683199

SCHEMBL9683199

FC(F)(F)c1ccc2c(c1)c(N1CCNCC1)nn2-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.51
HTR2C P28335 2/20 0.51
HTR3E A5X5Y0 2/20 0.51
HTR3B O95264 2/20 0.51
HTR3A P46098 2/20 0.51
HTR3D Q70Z44 2/20 0.51
HTR3C Q8WXA8 2/20 0.51
SIGMAR1 Q99720 2/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.50
THRB P10828 1/20 0.50
KHK P50053 7/20 0.48
HRH4 Q9H3N8 1/20 0.47
ADRB2 P07550 2/20 0.44
NCF1 P14598 1/20 0.44
HTR6 P50406 2/20 0.43
ADRB1 P08588 3/20 0.43
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9682489 0.85 HTR6 (0.47) HTR1DHTR2CHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9680573 0.84 HTR6 (0.46) HTR1DHTR2CHTR3EHTR3BHTR3A
SCHEMBL9682532 0.84 KHK (0.51) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL9680678 0.81 KHK (0.51) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL2710715 0.81 KHK (0.54) HTR2CHTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL9681346 0.79 KHK (0.53) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL9681249 0.77 HTR1A (0.48) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9681244 0.77 KHK (0.57) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9680691 0.74 KHK (0.57) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9681273 0.74 KHK (0.57) HTR2CHTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed