SCHEMBL9683181

SCHEMBL9683181

COc1ccc2c(N3CCNCC3)nn(-c3ccc(F)cc3)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 8/20 0.57
ADRB1 P08588 3/20 0.47
HTR3E A5X5Y0 2/20 0.47
HTR3B O95264 2/20 0.47
HTR3A P46098 2/20 0.47
HTR3D Q70Z44 2/20 0.47
HTR3C Q8WXA8 2/20 0.47
SIGMAR1 Q99720 1/20 0.47
HTR1A P08908 1/20 0.46
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NCF1 P14598 1/20 0.42
CYP1A2 P05177 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP1 P29466 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681919 0.91 KHK (0.52) KHKADRB1HTR3EHTR3BHTR3A
SCHEMBL9683240 0.87 KHK (0.50) KHKHTR1A
SCHEMBL9681219 0.81 KHK (0.56) KHKADRB1HTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9681291 0.80 KHK (0.55) KHKADRB1HTR3EHTR3BHTR3A
SCHEMBL9681244 0.80 KHK (0.57) KHKADRB1HTR3EHTR3BHTR3A
SCHEMBL9681305 0.79 KHK (0.47) KHKHTR3AHTR1AKDM4EMAPT
SCHEMBL9682300 0.75 GRIA1 (0.42) KHKHTR1AALDH1A1KDM4EHPGD
SCHEMBL9682530 0.74 KHK (0.51) KHKHTR3EHTR3BHTR3AHTR3D
SCHEMBL16712543 0.73 KHK (1.00) KHK
SCHEMBL9682532 0.72 KHK (0.51) KHKADRB1HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed