SCHEMBL9683256

SCHEMBL9683256

COc1cc[c]c(C(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
CYP2A6 P11509 1/20 0.39
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA7 P43166 3/20 0.35
CA9 Q16790 3/20 0.35
CA12 O43570 2/20 0.35
CA14 Q9ULX7 2/20 0.35
TAAR1 Q96RJ0 2/20 0.35
ALDH1A1 P00352 2/20 0.35
ACHE P22303 1/20 0.34
CYP2D6 P10635 2/20 0.34
RAB9A P51151 1/20 0.34
HTT P42858 1/20 0.34
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
CCR8 P51685 1/20 0.33
ABCB11 O95342 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7234655 0.84 TAAR1 (0.41) TAAR1ALDH1A1CYP2D6ABCB11CYP3A4
SCHEMBL11416597 0.82
SCHEMBL1078010 0.82 CA1 (0.34) CYP1A2CYP2A6CA1CA2CA7
SCHEMBL7482706 0.81 ABCB11 (0.37) TAAR1ALDH1A1ABCB11HTR2A
SCHEMBL27999512 0.77 PDE2A (0.37) CYP1A2ALDH1A1RAB9ACYP3A4
SCHEMBL11567095 0.76 CA4 (0.39) CYP1A2CYP2A6ALDH1A1
SCHEMBL10990313 0.75 MMP13 (0.33) ABCB11HTR2A
SCHEMBL15066961 0.73 ALDH1A1 (0.41) CYP1A2CYP2A6CA1CA2CA7
SCHEMBL4573904 0.73 ALDH1A1 (0.48) CYP1A2CYP2A6CA1CA2CA7
SCHEMBL15352571 0.72 NPSR1 (0.37) CYP1A2CYP2A6CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106573931-A Bet-protein inhibiting 3,4-dihydropyrido[2,3-b]pyrazinones with meta-substituted aromatic amino- or ether groups 拜耳医药股份有限公司 2017-04-19 CN disclosed
US-5169958-A Reacting, 3-amino-2-propen-1-ones with magnesium halide in solvent BASF AKTIENGESELLSCHAFT (DE) 1992-12-08 US disclosed
EP-0480242-A2 Method for the production of alpha,beta-unsaturated carbonyl compounds BASF Aktiengesellschaft (DE) 1992-04-15 EP disclosed
US-4578106-A Herbicidal esters of 2-bromo-4-methylimidazole-5-carboxylic acid STAUFFER CHEMICAL COMPANY (US) 1986-03-25 US disclosed
US-4129587-A ACRYLONITRILE WITH ORGANIC PHOSPHINITES OR PHOSPHONITES AS CATALYSTS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1978-12-12 US disclosed