Bumetrizole

Bumetrizole

SCHEMBL9683667

CCCCCCCCCCCCCCCCCCC(Cc1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1)C(=O)O.Cc1cc(-n2nc3ccc(Cl)cc3n2)c(O)c(C(C)(C)C)c1

nearest known ligand 0.35

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
PPARG P37231 6/20 0.33
PTGES O14684 1/20 0.33
ALOX5 P09917 1/20 0.33
CNR1 P21554 4/20 0.32
CNR2 P34972 4/20 0.32
KCNH2 Q12809 1/20 0.32
PPARA Q07869 8/20 0.31
POLB P06746 1/20 0.31
PPARD Q03181 4/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
MMP12 P39900 1/20 0.31
HMGCR P04035 1/20 0.30
F2R P25116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL224451 0.94 PPARG (0.35) PPARGPTGESALOX5CNR1CNR2
SCHEMBL15008371 0.87 PSEN1 (0.34) ALOX5CNR1CNR2MAPTHMGCR
Bumetrizole SCHEMBL8164248 0.84 NPC1 (0.40) NPC1RAB9APOLB
Bumetrizole SCHEMBL11754863 0.84 FFAR4 (0.40) NPC1RAB9A
SCHEMBL547105 0.84 PTGES (0.41) NPC1RAB9APPARGPTGESALOX5
SCHEMBL208254 0.84 MMP2 (0.33) PPARGPTGESALOX5MMP2
SCHEMBL208252 0.83 PPARG (0.31) PPARGCNR1CNR2PPARAPPARD
Bumetrizole SCHEMBL8379731 0.81 NPC1 (0.42) NPC1RAB9ACNR1CNR2POLB
Bumetrizole SCHEMBL11761050 0.81 NPC1 (0.35) NPC1RAB9APOLBHMGCR
Bumetrizole SCHEMBL3834201 0.81 NPC1 (0.45) NPC1RAB9APOLBTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124456-A HINDERED AMINE-SUBSTITUTED DIHYDROPYRIDINES AND HEAT/LIGHT STABILIZATION OF POLYMER SUBSTRATES THEREWITH RHONE-POULENC CHIMIE (FR) 1992-06-23 US disclosed