SCHEMBL9684893

SCHEMBL9684893

NC(=O)c1ccc(CCN(C[C@H](O)COc2ccccc2)C[C@H](O)COc2ccccc2)s1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
MAPT P10636 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
POLB P06746 1/20 0.44
GAA P10253 4/20 0.40
MAPK1 P28482 1/20 0.40
ABCB1 P08183 3/20 0.40
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TSHR P16473 2/20 0.38
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9684886 1.00 ALDH1A1 (0.47) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL9684099 0.83 ABCB1 (0.42) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL9684091 0.83 ABCB1 (0.42) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL9787435 0.80 ABCB1 (0.46) CYP2D6POLBGAAABCB1LMNA
SCHEMBL9787439 0.80 ABCB1 (0.46) CYP2D6POLBGAAABCB1LMNA
SCHEMBL10822432 0.80 KDM4E (0.44) ALDH1A1MEN1KMT2A
SCHEMBL10822435 0.80 KDM4E (0.44) ALDH1A1MEN1KMT2A
SCHEMBL10822438 0.80 KDM4E (0.44) ALDH1A1MEN1KMT2A
SCHEMBL9685069 0.80 ADRB1 (0.54) CYP1A2MEN1KMT2A
SCHEMBL9685064 0.80 ADRB1 (0.54) CYP1A2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166218-A Antilipemic agents or antiglycemic agents HOFFMANN-LA ROCHE INC. (US) 1992-11-24 US disclosed
US-5064863-A Catabolic activity, obesity, diabetes HOFFMANN-LA ROCHE INC. (US) 1991-11-12 US disclosed