SCHEMBL9685314

SCHEMBL9685314

Cc1ccc(-c2cccc(C#N)c2N)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.44
ADORA2A P29274 3/20 0.43
ADORA1 P30542 2/20 0.43
LRRK2 Q5S007 1/20 0.40
TSHR P16473 1/20 0.39
AR P10275 2/20 0.39
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 3/20 0.38
NPSR1 Q6W5P4 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP2A6 P11509 1/20 0.38
HPGD P15428 2/20 0.37
PPARG P37231 1/20 0.37
NCOA2 Q15596 1/20 0.37
NCOA1 Q15788 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27930441 0.85 ESR2 (0.47) ESR2TSHRARALDH1A1KDM4E
SCHEMBL28073082 0.84 LRRK2 (0.40) ESR2ADORA2AADORA1LRRK2TSHR
SCHEMBL27693511 0.83 ESR2 (0.48) ESR2ADORA2AADORA1LRRK2TSHR
SCHEMBL28367275 0.82 ALDH1A1 (0.57) ADORA2AADORA1ALDH1A1CYP2A6
SCHEMBL17940720 0.81 AR (0.42) ESR2LRRK2TSHRARALDH1A1
SCHEMBL7689092 0.81 POLB (0.49) ESR2ADORA2AADORA1TSHRAR
SCHEMBL29642877 0.81 AR (0.42) ESR2LRRK2TSHRARALDH1A1
SCHEMBL29799042 0.81 ESR2 (0.66) ESR2ADORA2AADORA1LRRK2TSHR
SCHEMBL27963955 0.81 ESR2 (0.66) ESR2ADORA2AADORA1LRRK2TSHR
SCHEMBL313 0.81 ESR2 (0.66) ESR2ADORA2AADORA1LRRK2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113228318-A Thermoelectric conversion material and thermoelectric conversion element using same 东洋油墨SC控股株式会社 2021-08-06 CN disclosed
EP-0245053-B1 HETEROCYCLIC FUSED TRICYCLIC COMPOUNDS ICI AMERICAS INC. (US) 1992-11-25 EP disclosed
US-5118688-A TETRAHYDROPYRIDOQUINOLONE DERIVATIVES USEFUL AS ANXIOLYTIC AGENTS ICI AMERICAS INC. (US) 1992-06-02 US disclosed
US-4975435-A Certain 1H-pyrrold[3,4-b]quinolin-1-one-9-amino-2,3-dihydro derivatives useful for treating anxiety ICI AMERICAS INC. (US) 1990-12-04 US disclosed
EP-0245053-A1 Heterocyclic fused tricyclic compounds ICI AMERICAS INC. (US) 1987-11-11 EP disclosed