SCHEMBL9685442

SCHEMBL9685442

CCOC1=CC(=O)NCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.38
LMNA P02545 1/20 0.33
CRBN Q96SW2 1/20 0.32
PARP1 P09874 1/20 0.31
ABCC4 O15439 1/20 0.31
ABCB11 O95342 1/20 0.31
CHRM2 P08172 1/20 0.31
ADRA2A P08913 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
CHRM1 P11229 1/20 0.31
ACHE P22303 1/20 0.31
PTGS1 P23219 1/20 0.31
PDE4A P27815 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31
CCNT1 O60563 1/20 0.30
CDK9 P50750 1/20 0.30
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3103319 0.89 PARP1 (0.38) HTTLMNAPARP1MEN1KMT2A
SCHEMBL31680983 0.87 FKBP5 (0.36) HTTLMNACRBNPARP1MEN1
SCHEMBL7770871 0.80
SCHEMBL1184 0.78
SCHEMBL1021859 0.71
SCHEMBL13469214 0.69
SCHEMBL99907 0.68 KMT2A (0.49) LMNAMEN1KMT2APOLB
SCHEMBL6515435 0.68 MEN1 (0.45) LMNAMEN1KMT2A
SCHEMBL2778609 0.68 MAPT (0.41) LMNAMEN1KMT2APOLBPLK4
SCHEMBL28957609 0.67 PGR (0.37) HTTLMNAKMT2APIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116554167-B Deuterated indolone derivative and application thereof in medicine 成都百裕制药股份有限公司 2024-06-25 CN disclosed
CN-116554167-A Deuterated indolone derivative and application thereof in medicine 成都百裕制药股份有限公司 2023-08-08 CN disclosed
US-9977024-B2 Targeted covalent probes and inhibitors of proteins containing redox-sensitive cysteines THE SCRIPPS RESEARCH INSTITUTE (US) 2018-05-22 US disclosed
EP-0245053-B1 HETEROCYCLIC FUSED TRICYCLIC COMPOUNDS ICI AMERICAS INC. (US) 1992-11-25 EP disclosed
US-5118688-A TETRAHYDROPYRIDOQUINOLONE DERIVATIVES USEFUL AS ANXIOLYTIC AGENTS ICI AMERICAS INC. (US) 1992-06-02 US disclosed
US-4975435-A Certain 1H-pyrrold[3,4-b]quinolin-1-one-9-amino-2,3-dihydro derivatives useful for treating anxiety ICI AMERICAS INC. (US) 1990-12-04 US disclosed
EP-0245053-A1 Heterocyclic fused tricyclic compounds ICI AMERICAS INC. (US) 1987-11-11 EP disclosed