SCHEMBL9686043

SCHEMBL9686043

O=P(O)(O)COCC1CCC(n2cnc3c(NC4CC4)ncnc32)C1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NT5E P21589 3/20 0.49
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49
ADORA1 P30542 2/20 0.46
GPR17 Q13304 1/20 0.45
ADCY5 O95622 5/20 0.45
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
P2RY1 P47900 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686090 0.84 ADCY5 (0.47) NT5EADCY5P2RY1
SCHEMBL9685235 0.84 ADCY5 (0.64) ADORA1ADCY5ADORA3
SCHEMBL9704183 0.83 ADORA3 (0.55) ADORA1ADORA3
SCHEMBL9704176 0.83 YTHDC1 (0.49) ADCY5ADORA3
SCHEMBL21839481 0.79 NT5E (0.77) NT5ETAS1R3TAS1R1ADORA1GPR17
SCHEMBL30394506 0.79 NT5E (0.77) NT5ETAS1R3TAS1R1ADORA1GPR17
SCHEMBL21883307 0.77 TAS1R3 (0.60) NT5ETAS1R3TAS1R1ADORA1GPR17
SCHEMBL9686031 0.77 ADORA3 (0.47) TAS1R3TAS1R1ADORA1CCNA2CDK2
SCHEMBL21883308 0.77 TAS1R3 (0.61) NT5ETAS1R3TAS1R1ADORA1GPR17
SCHEMBL21839754 0.75 TAS1R3 (0.81) NT5ETAS1R3TAS1R1ADORA1GPR17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468866-A1 Novel carbocyclic analogs of certain nucleosides MERRELL DOW PHARMACEUTICALS INC. (US) 1992-01-29 EP disclosed
EP-0468119-A1 Novel carbocyclic analogs of certain nucleosides MERRELL DOW PHARMACEUTICALS INC. (US) 1992-01-29 EP disclosed