SCHEMBL9686162

SCHEMBL9686162

C=Cc1ccc(N(C)C)cc1[N+](=O)[O-]

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.66
ACHE P22303 5/20 0.61
BCHE P06276 2/20 0.59
MAPT P10636 4/20 0.57
BACE1 P56817 4/20 0.53
NPSR1 Q6W5P4 1/20 0.51
ALDH1A1 P00352 2/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1647170 0.86 PTGS2 (0.66) PTGS2ACHEBCHEMAPTBACE1
SCHEMBL29559360 0.83 PTGS2 (0.71) PTGS2ACHEBCHEMAPTBACE1
SCHEMBL11795154 0.81 PTGS2 (0.63) PTGS2ACHEBCHEMAPTBACE1
SCHEMBL11795164 0.81 PTGS2 (0.63) PTGS2ACHEBCHEMAPTBACE1
SCHEMBL31361989 0.80 MAPT (0.72) PTGS2ACHEBCHEMAPTBACE1
SCHEMBL366120 0.79 TSHR (0.60) PTGS2ACHEMAPTNPSR1ALDH1A1
SCHEMBL9507521 0.79 MAPT (0.61) PTGS2ACHEBCHEMAPTBACE1
SCHEMBL10430142 0.79 PTGS2 (0.64) PTGS2ACHEBCHEMAPTBACE1
SCHEMBL1650914 0.79 PTGS2 (0.82) PTGS2ACHEBCHEMAPTBACE1
SCHEMBL1650911 0.79 PTGS2 (0.82) PTGS2ACHEBCHEMAPTBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0489547-A1 A process for the preparation of a 3-alkylated indole, intermediates, and a process for the preparation of a derivative thereof ZENECA LIMITED (GB) 1992-06-10 EP disclosed