SCHEMBL9686633

SCHEMBL9686633

CCN1CCc2nc(N3CCNCC3)ncc2C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.42
CYP1A2 P05177 13/20 0.42
HSD17B10 Q99714 13/20 0.42
CASP1 P29466 12/20 0.42
CASP7 P55210 12/20 0.42
HPGD P15428 10/20 0.42
CYP3A4 P08684 5/20 0.42
CYP2C19 P33261 4/20 0.42
TSHR P16473 3/20 0.42
CYP2C9 P11712 6/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CCNT1 O60563 1/20 0.41
CDK4 P11802 1/20 0.41
CCNA2 P20248 1/20 0.41
CCND1 P24385 1/20 0.41
CDK2 P24941 1/20 0.41
CCND3 P30281 1/20 0.41
CDK7 P50613 1/20 0.41
CDK9 P50750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1844326 0.89 ALDH1A1 (0.43) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL9686640 0.81 ALDH1A1 (0.44) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL9685453 0.80 ALDH1A1 (0.42) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL1921498 0.80 ALDH1A1 (0.42) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL9684514 0.78 LMNA (0.67) ALDH1A1HSD17B10HPGDTSHRUSP2
SCHEMBL22336033 0.77 HTR1A (0.49) MEN1KMT2AMAPTHTT
SCHEMBL1849473 0.76 ALDH1A1 (0.48) ALDH1A1CYP1A2HSD17B10CASP1CASP7
Hydrochloric Acid SCHEMBL31633382 0.76 USP2 (0.53) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL23282512 0.75 OGA (0.48) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL9685190 0.75 USP2 (0.66) ALDH1A1CYP1A2HSD17B10CASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
EP-0192783-B1 2-PIPERAZINOPYRIMIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1991-04-17 EP disclosed
US-4742165-A HERBICIDES MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-05-03 US disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0192783-A1 2-PIPERAZINOPYRIMIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-09-03 EP disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed