SCHEMBL9686635

SCHEMBL9686635

CC(C)Cc1cccc(C#N)c1N

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.46
GABRB2 P47870 1/20 0.46
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
ALOX5AP P20292 1/20 0.36
TSHR P16473 4/20 0.35
RORC P51449 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPK1 P28482 1/20 0.34
PLAU P00749 1/20 0.34
MAP2K1 Q02750 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA2 P47869 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isobutane SCHEMBL28311933 0.82 TSHR (0.35) SLC6A2SLC6A4ALOX5APTSHRKDM4E
SCHEMBL2659054 0.81 GABRA1 (0.47) GABRA1GABRB2SLC6A2SLC6A4ALOX5AP
SCHEMBL3960659 0.80 GABRA1 (0.60) GABRA1GABRB2SLC6A2SLC6A4GABRG2
SCHEMBL7863918 0.79 GABRA1 (0.40) GABRA1GABRB2TSHRKDM4EALDH1A1
SCHEMBL14983825 0.79 GABRA1 (0.46) GABRA1GABRB2SLC6A2SLC6A4ALOX5AP
SCHEMBL26463373 0.77 PNMT (0.39) TSHRKDM4EALDH1A1SMN1; SMN2PLAU
SCHEMBL6457244 0.76 AR (0.39) TSHRKDM4EALDH1A1HPGDMAPK1
SCHEMBL7806420 0.76 PDK2 (0.35) KDM4EALDH1A1PLAU
SCHEMBL9685552 0.76 CHRNE (0.37) TSHRKDM4EALDH1A1SMN1; SMN2PLAU
SCHEMBL10798754 0.76 PLAU (0.36) TSHRKDM4EALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0245053-B1 HETEROCYCLIC FUSED TRICYCLIC COMPOUNDS ICI AMERICAS INC. (US) 1992-11-25 EP disclosed
US-5118688-A TETRAHYDROPYRIDOQUINOLONE DERIVATIVES USEFUL AS ANXIOLYTIC AGENTS ICI AMERICAS INC. (US) 1992-06-02 US disclosed
US-4975435-A Certain 1H-pyrrold[3,4-b]quinolin-1-one-9-amino-2,3-dihydro derivatives useful for treating anxiety ICI AMERICAS INC. (US) 1990-12-04 US disclosed
EP-0245053-A1 Heterocyclic fused tricyclic compounds ICI AMERICAS INC. (US) 1987-11-11 EP disclosed