SCHEMBL9685552

SCHEMBL9685552

N#Cc1cccc(CO)c1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNE Q04844 1/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PLAU P00749 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ESR2 Q92731 1/20 0.36
MAP2K1 Q02750 1/20 0.36
KDM4E B2RXH2 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
TSHR P16473 1/20 0.34
CYP19A1 P11511 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
LMNA P02545 1/20 0.33
GALR3 O60755 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL84271 0.85 PLAU (0.35) ALDH1A1MAPTSMN1; SMN2PLAUESR2
SCHEMBL26463373 0.82 PNMT (0.39) ALDH1A1MAPTSMN1; SMN2PLAUCA1
SCHEMBL7863918 0.80 GABRA1 (0.40) ALDH1A1MAPTPLAUCA1CA2
SCHEMBL10798754 0.80 PLAU (0.36) ALDH1A1MAPTSMN1; SMN2PLAUCA1
SCHEMBL483697 0.79 ALDH1A1 (0.49) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL30496165 0.79 ALDH1A1 (0.49) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL15390567 0.78 APOBEC3G (0.44) CHRNEALDH1A1MAPTKDM4ECYP3A4
SCHEMBL2423501 0.78 TSHR (0.46) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL1378624 0.78 CA1 (0.41) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL28215006 0.78 S1PR1 (0.40) ALDH1A1MAPTSMN1; SMN2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0245053-B1 HETEROCYCLIC FUSED TRICYCLIC COMPOUNDS ICI AMERICAS INC. (US) 1992-11-25 EP disclosed
US-5118688-A TETRAHYDROPYRIDOQUINOLONE DERIVATIVES USEFUL AS ANXIOLYTIC AGENTS ICI AMERICAS INC. (US) 1992-06-02 US disclosed
US-4975435-A Certain 1H-pyrrold[3,4-b]quinolin-1-one-9-amino-2,3-dihydro derivatives useful for treating anxiety ICI AMERICAS INC. (US) 1990-12-04 US disclosed
EP-0245053-A1 Heterocyclic fused tricyclic compounds ICI AMERICAS INC. (US) 1987-11-11 EP disclosed