SCHEMBL9686831

SCHEMBL9686831

C=CCN1CC(=O)C(C(=O)OCC)C1=O

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
MAPT P10636 2/20 0.34
TLR4 O00206 1/20 0.33
ELANE P08246 1/20 0.33
CTSG P08311 1/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685183 0.81 ALDH1A1 (0.42) ALDH1A1MAPTTLR4POLBLMNA
SCHEMBL10366484 0.78 ALDH1A1 (0.49) ALDH1A1MAPTTLR4POLBKMT2A
SCHEMBL3367604 0.73 ALDH1A1 (0.39) ALDH1A1MAPTTLR4KMT2AKDM4E
SCHEMBL10367891 0.72 MAPT (0.38) ALDH1A1MAPTPOLBLMNAKMT2A
SCHEMBL9685715 0.72 POLB (0.39) ALDH1A1MAPTTLR4POLBKMT2A
SCHEMBL22216178 0.72 MAPT (0.52) ALDH1A1MAPTTLR4POLBKMT2A
SCHEMBL22715440 0.71 ALDH1A1 (0.61) ALDH1A1MAPTTLR4ELANECTSG
SCHEMBL9042858 0.70 ALDH1A1 (0.60) ALDH1A1MAPTLMNAKMT2AKDM4E
SCHEMBL11732751 0.69 ALDH1A1 (0.40) ALDH1A1MAPTTLR4ELANECTSG
SCHEMBL22216464 0.69 MAPT (0.40) ALDH1A1MAPTTLR4LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0245053-B1 HETEROCYCLIC FUSED TRICYCLIC COMPOUNDS ICI AMERICAS INC. (US) 1992-11-25 EP disclosed
US-5118688-A TETRAHYDROPYRIDOQUINOLONE DERIVATIVES USEFUL AS ANXIOLYTIC AGENTS ICI AMERICAS INC. (US) 1992-06-02 US disclosed
US-4975435-A Certain 1H-pyrrold[3,4-b]quinolin-1-one-9-amino-2,3-dihydro derivatives useful for treating anxiety ICI AMERICAS INC. (US) 1990-12-04 US disclosed
EP-0178759-B1 ALKYNYL DERIVATIVESOF PYRAZOLO-(3,4-B)-PYRIDINE LACTAMS ICI AMERICAS INC. (US) 1990-01-10 EP disclosed
EP-0245053-A1 Heterocyclic fused tricyclic compounds ICI AMERICAS INC. (US) 1987-11-11 EP disclosed
US-4705793-A Pyrazolo[3,4-b]pyrrolo[3,4-e]pyridine-5(1H)-one and 1-H-pyrazolo[3,4-b][1,6]naphthyridine-5(6H)-one derivations, useful as anti-anxiety agents ICI AMERICAS INC. (US) 1987-11-10 US disclosed
EP-0178759-A1 Alkynyl derivativesof pyrazolo-(3,4-b)-pyridine lactams ICI AMERICAS INC. (US) 1986-04-23 EP disclosed