SCHEMBL9685183

SCHEMBL9685183

CCCN1CC(=O)C(C(=O)OCC)C1=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
MAPT P10636 3/20 0.36
TLR4 O00206 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
POLB P06746 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
FKBP1A P62942 1/20 0.34
HTT P42858 2/20 0.33
LMNA P02545 1/20 0.33
PARP1 P09874 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10366484 0.91 ALDH1A1 (0.49) ALDH1A1MAPTTLR4KDM4EMEN1
SCHEMBL10749202 0.87 FKBP1A (0.44) ALDH1A1MAPTKDM4EL3MBTL1FKBP1A
SCHEMBL9686831 0.81 ALDH1A1 (0.34) ALDH1A1MAPTTLR4KDM4EMEN1
SCHEMBL3367604 0.76 ALDH1A1 (0.39) ALDH1A1MAPTTLR4KDM4EMEN1
SCHEMBL9685715 0.75 POLB (0.39) ALDH1A1MAPTTLR4KDM4EMEN1
SCHEMBL22216178 0.75 MAPT (0.52) ALDH1A1MAPTTLR4KDM4EMEN1
SCHEMBL1303947 0.74 ALDH1A1 (0.39) ALDH1A1MAPTTLR4KDM4EMEN1
SCHEMBL22206975 0.74 ALDH1A1 (0.39) ALDH1A1MAPTKDM4EGAAHPGD
SCHEMBL9042858 0.73 ALDH1A1 (0.60) ALDH1A1MAPTKDM4EMEN1GAA
SCHEMBL7009722 0.72 BRD4 (0.38) ALDH1A1MAPTKMT2AFKBP1ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0245053-B1 HETEROCYCLIC FUSED TRICYCLIC COMPOUNDS ICI AMERICAS INC. (US) 1992-11-25 EP disclosed
US-5118688-A TETRAHYDROPYRIDOQUINOLONE DERIVATIVES USEFUL AS ANXIOLYTIC AGENTS ICI AMERICAS INC. (US) 1992-06-02 US disclosed
US-4975435-A Certain 1H-pyrrold[3,4-b]quinolin-1-one-9-amino-2,3-dihydro derivatives useful for treating anxiety ICI AMERICAS INC. (US) 1990-12-04 US disclosed
EP-0178759-B1 ALKYNYL DERIVATIVESOF PYRAZOLO-(3,4-B)-PYRIDINE LACTAMS ICI AMERICAS INC. (US) 1990-01-10 EP disclosed
EP-0245053-A1 Heterocyclic fused tricyclic compounds ICI AMERICAS INC. (US) 1987-11-11 EP disclosed
US-4705793-A Pyrazolo[3,4-b]pyrrolo[3,4-e]pyridine-5(1H)-one and 1-H-pyrazolo[3,4-b][1,6]naphthyridine-5(6H)-one derivations, useful as anti-anxiety agents ICI AMERICAS INC. (US) 1987-11-10 US disclosed
EP-0178759-A1 Alkynyl derivativesof pyrazolo-(3,4-b)-pyridine lactams ICI AMERICAS INC. (US) 1986-04-23 EP disclosed