SCHEMBL9687085

SCHEMBL9687085

O=C1CCCc2c1c(-c1ccccc1)nn2-c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.66
PTGS1 P23219 6/20 0.61
ALDH1A1 P00352 3/20 0.51
MAPK10 P53779 1/20 0.51
SRC P12931 1/20 0.47
HPGD P15428 3/20 0.47
KMT2A Q03164 3/20 0.47
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 2/20 0.47
LMNA P02545 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HTT P42858 2/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CSNK2B P67870 1/20 0.45
CSNK2A1 P68400 1/20 0.45
MAPT P10636 2/20 0.43
TSHR P16473 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6162529 0.83 OPRM1 (0.56) PTGS2ALDH1A1MAPK10SRCHPGD
SCHEMBL6166055 0.79 ALDH1A1 (0.46) PTGS2PTGS1ALDH1A1MAPK10SRC
SCHEMBL6167303 0.78 ALDH1A1 (0.45) PTGS2PTGS1ALDH1A1MAPK10SRC
SCHEMBL6165988 0.78 ALDH1A1 (0.45) PTGS2PTGS1ALDH1A1MAPK10SRC
SCHEMBL6165127 0.78 ALDH1A1 (0.43) PTGS2PTGS1ALDH1A1MAPK10SRC
SCHEMBL5698532 0.78 PTGS2 (0.64) PTGS2PTGS1ALDH1A1MAPK10SRC
SCHEMBL6162867 0.76 ALDH1A1 (0.49) PTGS2PTGS1ALDH1A1MAPK10SRC
SCHEMBL16516850 0.71 ALDH1A1 (0.41) PTGS2ALDH1A1MAPK10SRCHPGD
SCHEMBL23657754 0.70 PTGS1 (0.47) PTGS2PTGS1ALDH1A1HPGDKMT2A
SCHEMBL6163485 0.70 ALDH1A1 (0.38) PTGS2PTGS1ALDH1A1MAPK10SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5079258-A Enzyme inhibitors, antiallergens treatment of asthma BAYER AKTIENGESELLSCHAFT (DE) 1992-01-07 US claimed
US-5104442-A Cereals HOECHST AKTIENGESELLSCHAFT (DE) 1992-04-14 US disclosed
EP-0470489-A1 4,5,6,7-Tetrahydro-3-aryl-indazoles, process for their preparation and their use as herbicides HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-12 EP disclosed