SCHEMBL9687973

SCHEMBL9687973

[CH](c1ccccn1)c1nc2ccccc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 1/20 0.56
RAB9A P51151 14/20 0.54
NPC1 O15118 13/20 0.54
MAPT P10636 7/20 0.54
PKM P14618 6/20 0.54
GAA P10253 4/20 0.54
HTT P42858 4/20 0.54
NPSR1 Q6W5P4 3/20 0.54
ALDH1A1 P00352 9/20 0.50
SMN1; SMN2 Q16637 8/20 0.50
KMT2A Q03164 8/20 0.50
HPGD P15428 7/20 0.50
MEN1 O00255 7/20 0.50
KDM4E B2RXH2 7/20 0.50
LMNA P02545 6/20 0.50
MTOR P42345 1/20 0.50
METAP2 P50579 1/20 0.50
METAP1 P53582 1/20 0.50
HSP90AA1 P07900 1/20 0.50
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL709071 0.87 NPC1 (0.64) FGFR1RAB9ANPC1MAPTPKM
SCHEMBL709072 0.87 NPC1 (0.64) FGFR1RAB9ANPC1MAPTPKM
SCHEMBL19119423 0.82 ALDH1A1 (0.63) RAB9ANPC1MAPTPKMGAA
SCHEMBL1086985 0.74 ALDH1A1 (0.81) RAB9ANPC1MAPTPKMGAA
SCHEMBL1086983 0.74 ALDH1A1 (0.81) RAB9ANPC1MAPTPKMGAA
SCHEMBL29539476 0.74 ALDH1A1 (0.81) RAB9ANPC1MAPTPKMGAA
Quinoline SCHEMBL27617889 0.71 ALDH1A1 (0.53) FGFR1RAB9ANPC1MAPTPKM
SCHEMBL41190 0.71 RAB9A (0.74) RAB9ANPC1PKMALDH1A1KMT2A
SCHEMBL3081168 0.71 ALDH1A1 (0.59) RAB9ANPC1MAPTPKMGAA
SCHEMBL376644 0.71 ALDH1A1 (0.59) RAB9ANPC1MAPTPKMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201575-B1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1992-08-12 EP claimed
EP-0166287-B1 DIALKOXYRIDINES, PROCESS FOR THEIR PREPARATION, THEIR APPLICATION AND MEDICAMENTS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1989-08-23 EP claimed
US-4686230-A Picoline derivative useful as gastric acid secretion inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1987-08-11 US disclosed