SCHEMBL9688697

SCHEMBL9688697

CCC(Cc1nnc(S)n1C)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
CA2 P00918 1/20 0.34
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 2/20 0.34
CYP1A2 P05177 2/20 0.33
CHRM1 P11229 2/20 0.33
ADRA1A P35348 2/20 0.33
TBXA2R P21731 1/20 0.33
PDE4A P27815 1/20 0.33
LMNA P02545 1/20 0.33
CYP2C9 P11712 1/20 0.33
HIF1A Q16665 1/20 0.33
SLC1A3 P43003 1/20 0.33
SLC1A2 P43004 1/20 0.33
SLC1A1 P43005 1/20 0.33
NR4A2 P43354 1/20 0.33
AKR1A1 P14550 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11314946 0.72 ALDH1A1 (0.33) MAPK1
SCHEMBL16312316 0.69 CYP1A2 (0.35) MAPK1CYP1A2LMNACYP2C9
SCHEMBL11423451 0.66 KMT2A (0.34)
SCHEMBL13865681 0.63
SCHEMBL14112926 0.63
SCHEMBL6114 0.62
SCHEMBL16508860 0.61 CPB2 (0.51) CYP2C9
Hydrochloric Acid SCHEMBL2210811 0.60
SCHEMBL2355348 0.60
SCHEMBL8573707 0.60

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0329357-B1 DIHYDROPYRIDINE ANTI-ALLERGIC AND ANTI-INFLAMMATORY AGENTS Pfizer Limited (GB) 1992-07-15 EP disclosed
EP-0329357-A1 Dihydropyridine anti-allergic and anti-inflammatory agents Pfizer Limited (GB) 1989-08-23 EP disclosed
US-4859686-A Dihydropyridine anti-allergic and anti-inflammatory agents PFIZER INC. (US) 1989-08-22 US disclosed