SCHEMBL9688973

SCHEMBL9688973

COc1ccc(CCNC(=O)C(F)(F)F)c(C(=O)O)c1N

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.46
MTNR1B P49286 5/20 0.46
NQO2 P16083 2/20 0.41
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10410596 0.90 MTNR1A (0.46) MTNR1AMTNR1BNQO2ALDH1A1CYP1A2
SCHEMBL5076870 0.75 MTNR1A (0.68) MTNR1AMTNR1BALDH1A1
SCHEMBL27229064 0.74 MTNR1A (0.65) MTNR1AMTNR1BNQO2
SCHEMBL9786035 0.74 SLC2A1 (0.47) MTNR1AMTNR1BNQO2ALDH1A1
SCHEMBL5913864 0.73 CA12 (0.51)
SCHEMBL10409132 0.73 MTNR1A (0.41) MTNR1AMTNR1BNQO2
SCHEMBL18159090 0.72 NQO2 (0.49) MTNR1AMTNR1BNQO2
SCHEMBL27229027 0.72 MTNR1A (0.49) MTNR1AMTNR1BNQO2
SCHEMBL18159182 0.72 SMN1; SMN2 (0.52) MTNR1AMTNR1BNQO2ALDH1A1
SCHEMBL9688747 0.71 ALDH1A1 (0.51) MTNR1AMTNR1BNQO2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed
EP-0189473-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS. SCHERING AG (DE) 1986-08-06 EP disclosed
WO-1986001204-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1986-02-27 WO disclosed