SCHEMBL9689449

SCHEMBL9689449

COc1cc(CCNC(=O)C(F)(F)F)cc2c(=O)[nH][nH]c12

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.43
ALDH1A1 P00352 1/20 0.43
MTNR1B P49286 4/20 0.42
NQO2 P16083 2/20 0.40
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25179253 0.80 MTNR1A (0.46) MTNR1AMTNR1BNQO2
SCHEMBL9687908 0.80 MTNR1A (0.42) MTNR1AALDH1A1MTNR1BNQO2
SCHEMBL25186090 0.75 MTNR1A (0.46) MTNR1AALDH1A1MTNR1BNQO2
SCHEMBL1968355 0.75 CA12 (0.66) ALDH1A1
SCHEMBL9688747 0.74 ALDH1A1 (0.51) MTNR1AALDH1A1MTNR1BNQO2
SCHEMBL9689788 0.74 HTR2A (0.51)
SCHEMBL25198660 0.74 MTNR1A (0.46) MTNR1AMTNR1BNQO2
SCHEMBL25186468 0.74 MTNR1A (0.43) MTNR1AMTNR1BNQO2
SCHEMBL21693911 0.73 MEN1 (0.48)
SCHEMBL25183361 0.73 MTNR1A (0.45) MTNR1AALDH1A1MTNR1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed
EP-0189473-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS. SCHERING AG (DE) 1986-08-06 EP disclosed
WO-1986001204-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1986-02-27 WO disclosed