SCHEMBL9689495

SCHEMBL9689495

CCNc1cccnc1N1CCN(CCCCc2cc(C)c(O)c(C)c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
DRD2 P14416 7/20 0.41
DRD3 P35462 7/20 0.41
HTR1A P08908 5/20 0.41
HTR2A P28223 4/20 0.41
HTR7 P34969 4/20 0.41
HTR2C P28335 1/20 0.41
DRD1 P21728 2/20 0.41
DRD5 P21918 2/20 0.41
ADRA1A P35348 2/20 0.39
DRD4 P21917 4/20 0.39
ADRA2C P18825 1/20 0.39
HRH1 P35367 1/20 0.39
POLB P06746 1/20 0.38
CHIA Q9BZP6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9689294 0.99 PARP1 (0.41) PARP1DRD2DRD3HTR1AHTR2A
Hydrochloric Acid SCHEMBL10365165 0.99 PARP1 (0.41) PARP1DRD2DRD3HTR1AHTR2A
SCHEMBL9689578 0.97 PARP1 (0.42) PARP1DRD2DRD3HTR1AHTR2A
SCHEMBL9689955 0.93 PARP1 (0.43) PARP1DRD2DRD4CHIA
SCHEMBL9689504 0.88 HTR1A (0.45) PARP1DRD2DRD3HTR1AHTR2A
Hydrochloric Acid SCHEMBL9688128 0.87 HTR1A (0.44) PARP1DRD2DRD3HTR1AHTR2A
SCHEMBL9036531 0.86 PPARG (0.46) PARP1HTR1AHTR2CCHIA
SCHEMBL9689032 0.85 DRD2 (0.44) PARP1DRD2DRD3HTR1AHTR2A
SCHEMBL9689554 0.81 AURKA (0.40) PARP1DRD2DRD3HTR1AHTR2A
SCHEMBL9689528 0.81 PARP1 (0.47) PARP1DRD2DRD3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed