SCHEMBL9689504

SCHEMBL9689504

CCNc1cccnc1N1CCN(CCCCc2cc(C)c(OC)c(C)c2)CC1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.45
DRD2 P14416 8/20 0.42
DRD3 P35462 5/20 0.42
DRD4 P21917 1/20 0.42
HTR2A P28223 6/20 0.40
HTR7 P34969 5/20 0.40
DRD1 P21728 1/20 0.40
DRD5 P21918 1/20 0.40
ADRA1A P35348 3/20 0.39
PARP1 P09874 1/20 0.39
ELANE P08246 1/20 0.38
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9688128 0.99 HTR1A (0.44) HTR1ADRD2DRD3DRD4HTR2A
SCHEMBL9689032 0.97 DRD2 (0.44) HTR1ADRD2DRD3DRD4HTR2A
SCHEMBL9689554 0.93 AURKA (0.40) HTR1ADRD2DRD3DRD4HTR2A
Hydrochloric Acid SCHEMBL9704402 0.92 HTR2A (0.40) HTR1ADRD2DRD3DRD4HTR2A
SCHEMBL9689495 0.88 PARP1 (0.42) HTR1ADRD2DRD3DRD4HTR2A
Hydrochloric Acid SCHEMBL9689294 0.87 PARP1 (0.41) HTR1ADRD2DRD3DRD4HTR2A
Hydrochloric Acid SCHEMBL10365165 0.87 PARP1 (0.41) HTR1ADRD2DRD3DRD4HTR2A
SCHEMBL9037849 0.87 PPARG (0.48) HTR1ADRD2DRD3DRD4PARP1
Hydrochloric Acid SCHEMBL22150567 0.86 PPARG (0.48) HTR1ADRD2DRD3DRD4PARP1
SCHEMBL9689578 0.85 PARP1 (0.42) HTR1ADRD2DRD3DRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed