SCHEMBL9689517

SCHEMBL9689517

COc1cccc(CNC(CO)c2ccc(OC)c(OC)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
POLB P06746 1/20 0.50
ABCB1 P08183 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
CASR P41180 5/20 0.47
PPARA Q07869 2/20 0.47
KDM4E B2RXH2 1/20 0.46
PPARG P37231 1/20 0.46
PPARD Q03181 1/20 0.46
HDAC8 Q9BY41 1/20 0.45
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MMP13 P45452 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18114399 0.85 CASR (0.60) CASRMEN1KMT2A
SCHEMBL16463600 0.81 CASR (0.70) POLBCASRMEN1KMT2A
SCHEMBL8904970 0.79 OPRK1 (0.57) ALDH1A1POLBMEN1KMT2ALMNA
SCHEMBL28063503 0.78 PPARG (0.55) ALDH1A1POLBPPARAPPARGPPARD
SCHEMBL11041312 0.76 PKM (0.54) ALDH1A1PPARAKDM4EPPARGPPARD
SCHEMBL9585590 0.75 PPARG (0.53) ALDH1A1POLBPPARAPPARGPPARD
SCHEMBL8358298 0.75 CHRM2 (0.51) ALDH1A1POLBABCB1ABCG2HTT
SCHEMBL7324272 0.75 LMNA (0.47) ALDH1A1POLBCASRSMN1; SMN2MEN1
SCHEMBL4889095 0.74 POLB (0.62) ALDH1A1POLBSMN1; SMN2MEN1KMT2A
SCHEMBL4889036 0.74 POLB (0.62) ALDH1A1POLBSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed