SCHEMBL9689809

SCHEMBL9689809

c1ccc(CCN2CCC(Nc3nc4ccccc4[nH]3)C2)cc1

nearest known ligand 0.72

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.72
CHRNA7 P36544 1/20 0.49
GAA P10253 2/20 0.48
MAPT P10636 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
TP53 P04637 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
DNMT3A Q9Y6K1 1/20 0.47
GFER P55789 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
OPRK1 P41145 1/20 0.47
GRIN2B Q13224 2/20 0.46
GRIN1 Q05586 1/20 0.46
JAK1 P23458 1/20 0.46
PARP1 P09874 1/20 0.45
SSTR5 P35346 1/20 0.45
GRIN2A Q12879 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11266594 0.94 KCNH2 (0.80) KCNH2CHRNA7GAAMAPTL3MBTL1
SCHEMBL9689872 0.88 KCNH2 (0.90) KCNH2GAAMAPTL3MBTL1TP53
SCHEMBL1101038 0.85 KCNH2 (0.77) KCNH2CHRNA7DNMT3ASSTR5TSHR
SCHEMBL3748349 0.84 KCNH2 (0.63) KCNH2GAAMAPTL3MBTL1TP53
SCHEMBL9691007 0.84 KCNH2 (0.59) KCNH2RAB9A
SCHEMBL9538063 0.83 KCNH2 (1.00) KCNH2GAAMAPTL3MBTL1TP53
SCHEMBL9689110 0.81 KCNH2 (0.57) KCNH2CHRNA7GAAMAPTL3MBTL1
SCHEMBL9690409 0.81 KCNH2 (0.55) KCNH2CHRNA7GAARAB9ASMN1; SMN2
SCHEMBL662101 0.80 PARP1 (0.64) KCNH2CHRNA7GRIN2BGRIN1PARP1
SCHEMBL9698375 0.80 KCNH2 (0.66) KCNH2CHRNA7SMN1; SMN2GRIN2BJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed