SCHEMBL9690409

SCHEMBL9690409

c1cnc(NCCN2CCC(Nc3nc4ccccc4[nH]3)C2)nc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.55
TSHR P16473 1/20 0.51
CHRNA7 P36544 1/20 0.43
CXCR4 P61073 1/20 0.42
PDE10A Q9Y233 1/20 0.41
DRD4 P21917 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SLC40A1 Q9NP59 1/20 0.41
ERN1 O75460 1/20 0.40
MAPK10 P53779 1/20 0.40
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1151915 0.94 KCNH2 (0.59) KCNH2TSHRCHRNA7PDE10ADRD4
SCHEMBL8135558 0.82 KCNH2 (0.45) KCNH2TSHR
SCHEMBL9689809 0.81 KCNH2 (0.72) KCNH2TSHRCHRNA7GAARAB9A
SCHEMBL9691007 0.79 KCNH2 (0.59) KCNH2NPC1RAB9A
SCHEMBL10508648 0.79 KCNH2 (0.55) KCNH2TSHRCHRNA7PDE10ADRD4
SCHEMBL8562586 0.79 KCNH2 (0.65) KCNH2TSHRCHRNA7PDE10ADRD4
SCHEMBL9689110 0.77 KCNH2 (0.57) KCNH2TSHRCHRNA7GAA
SCHEMBL10749867 0.77 KCNH2 (0.59) KCNH2TSHRCHRNA7KDM4EGAA
Water SCHEMBL11093961 0.76 CXCR3 (0.51) KCNH2TSHRCHRNA7DRD4KDM4E
SCHEMBL11266594 0.76 KCNH2 (0.80) KCNH2TSHRCHRNA7GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed