SCHEMBL9689110

SCHEMBL9689110

S=C=NCCN1CCC(Nc2nc3ccccc3[nH]2)C1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.57
TSHR P16473 1/20 0.41
CHRNA7 P36544 1/20 0.40
USP30 Q70CQ3 2/20 0.40
KCNN3 Q9UGI6 2/20 0.39
HDAC6 Q9UBN7 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
GFER P55789 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KCNN1 Q92952 1/20 0.38
KCNN2 Q9H2S1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689809 0.81 KCNH2 (0.72) KCNH2TSHRCHRNA7GAAMAPT
SCHEMBL9536746 0.79 KCNH2 (0.46) KCNH2MAPT
SCHEMBL9690409 0.77 KCNH2 (0.55) KCNH2TSHRCHRNA7GAA
SCHEMBL9691007 0.77 KCNH2 (0.59) KCNH2
SCHEMBL11266594 0.76 KCNH2 (0.80) KCNH2TSHRCHRNA7GAAMAPT
SCHEMBL9689872 0.76 KCNH2 (0.90) KCNH2GAAMAPTL3MBTL1
SCHEMBL9698375 0.75 KCNH2 (0.66) KCNH2TSHRCHRNA7KCNN3HDAC6
SCHEMBL9697190 0.75 KCNH2 (0.66) KCNH2TSHRKCNN3HDAC6
SCHEMBL7416758 0.75 KCNH2 (0.65) KCNH2TSHRKCNN3HDAC6
SCHEMBL8560605 0.73 KCNH2 (0.61) KCNH2KCNN3HDAC6KCNN1KCNN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed