SCHEMBL9689831

SCHEMBL9689831

NC(=S)NCCN1CCC(Nc2nc3cccnc3n2Cc2cscn2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.36
TP53 P04637 4/20 0.35
EED O75530 2/20 0.35
SCN9A Q15858 1/20 0.34
KCNH2 Q12809 6/20 0.33
NR4A2 P43354 1/20 0.33
SSTR5 P35346 3/20 0.33
MAPT P10636 2/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
OPRM1 P35372 3/20 0.32
OPRD1 P41143 3/20 0.32
OPRK1 P41145 2/20 0.32
ENPP2 Q13822 1/20 0.32
SLC40A1 Q9NP59 1/20 0.31
MEN1 O00255 1/20 0.31
MLNR O43193 1/20 0.31
CACNA1F O60840 1/20 0.31
USP2 O75604 1/20 0.31
ABCB11 O95342 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9629392 0.90 TP53 (0.40) HTR1ATP53EEDSCN9AKCNH2
SCHEMBL9688923 0.89 EED (0.46) HTR1ATP53EEDKCNH2NR4A2
SCHEMBL9630461 0.88 HTR1A (0.40) HTR1ATP53EEDSCN9AKCNH2
SCHEMBL9629371 0.87 HTR1A (0.42) HTR1ATP53EEDSCN9AKCNH2
SCHEMBL9631303 0.86 ROCK2 (0.35) HTR1ATP53
SCHEMBL9691136 0.85 SLC6A9 (0.44) TP53EEDMAPTENPP2
SCHEMBL9630201 0.83 HTR1A (0.37) HTR1ATP53EEDSCN9AKCNH2
Fumaric Acid SCHEMBL9807334 0.82 HTR1A (0.37) HTR1ATP53EEDSCN9AKCNH2
SCHEMBL9690678 0.82 MEN1 (0.39) HTR1ATP53EEDKCNH2NR4A2
Oxalic Acid SCHEMBL9629056 0.79 CHEK2 (0.37) HTR1ASCN9AKCNH2MAPTFNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed