SCHEMBL9689854

SCHEMBL9689854

COC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1cc([N+](=O)[O-])ccc1OCCCCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.50
MAPT P10636 5/20 0.48
HIF1A Q16665 4/20 0.48
CYP1A2 P05177 4/20 0.48
CYP3A4 P08684 4/20 0.48
CYP2C9 P11712 4/20 0.48
CYP2C19 P33261 4/20 0.48
KMT2A Q03164 4/20 0.48
CYP2D6 P10635 3/20 0.48
ADORA3 P0DMS8 3/20 0.48
TDP1 Q9NUW8 3/20 0.48
LMNA P02545 2/20 0.48
TSHR P16473 2/20 0.48
NFKB1 P19838 2/20 0.48
MAPK1 P28482 2/20 0.48
THPO P40225 2/20 0.48
KCNK2 O95069 2/20 0.48
TP53 P04637 2/20 0.48
DRD1 P21728 2/20 0.48
HTR2C P28335 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691974 0.95 HSD17B10 (0.54) HSD17B10MAPTHIF1ACYP1A2CYP3A4
SCHEMBL9824964 0.87 CACNA1C (0.49) MAPTHIF1ACYP1A2CYP3A4CYP2C9
SCHEMBL10689136 0.85 HSD17B10 (0.51) HSD17B10MAPTHIF1ACYP1A2CYP3A4
SCHEMBL7287257 0.84 ADORA3 (0.53) HSD17B10MAPTHIF1ACYP1A2CYP3A4
SCHEMBL10488355 0.84 ADORA3 (0.53) HSD17B10MAPTHIF1ACYP1A2CYP3A4
SCHEMBL10922862 0.83 CACNA1C (0.52) HSD17B10MAPTHIF1ACYP1A2CYP3A4
SCHEMBL9789920 0.83 ADORA3 (0.52) HSD17B10MAPTHIF1ACYP1A2CYP3A4
SCHEMBL10488517 0.83 ADORA3 (0.53) HSD17B10MAPTHIF1ACYP1A2CYP3A4
SCHEMBL7347116 0.82 HSD17B10 (0.56) HSD17B10MAPTHIF1ACYP1A2CYP3A4
SCHEMBL9672729 0.82 CACNA1F (0.68) MAPTHIF1ACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0194751-B1 DIHYDROPYRIDINE ALKANOL AMINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-04-15 EP disclosed
US-4873254-A ADRENERGIC BLOCKING AGENTS OR CALCIUM CHANNEL BLOCKERS; HYPOTENSIVE AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-10-10 US disclosed
EP-0194047-A1 Dihydropyridine alkanol amines, process for their preparation and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-09-10 EP disclosed