SCHEMBL10691974

SCHEMBL10691974

COC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1cc([N+](=O)[O-])ccc1OCCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.54
LMNA P02545 3/20 0.51
ALDH1A1 P00352 2/20 0.51
AGTR1 P30556 2/20 0.51
RAB9A P51151 1/20 0.49
HIF1A Q16665 4/20 0.49
MAPT P10636 4/20 0.49
KMT2A Q03164 4/20 0.49
CYP1A2 P05177 3/20 0.49
CYP3A4 P08684 3/20 0.49
CYP2C9 P11712 3/20 0.49
CYP2C19 P33261 3/20 0.49
CYP2D6 P10635 2/20 0.49
TSHR P16473 2/20 0.49
NFKB1 P19838 2/20 0.49
MAPK1 P28482 2/20 0.49
THPO P40225 2/20 0.49
ADORA3 P0DMS8 2/20 0.49
CACNA1C Q13936 2/20 0.49
TDP1 Q9NUW8 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689854 0.95 HSD17B10 (0.50) HSD17B10LMNAALDH1A1AGTR1HIF1A
SCHEMBL7347116 0.85 HSD17B10 (0.56) HSD17B10LMNAHIF1AMAPTKMT2A
SCHEMBL10691979 0.84 LMNA (0.61) HSD17B10LMNAALDH1A1AGTR1RAB9A
SCHEMBL9825000 0.83 ADORA3 (0.54) HSD17B10LMNAALDH1A1AGTR1HIF1A
SCHEMBL10488517 0.82 ADORA3 (0.53) HSD17B10LMNAALDH1A1AGTR1HIF1A
SCHEMBL10692951 0.82 ADORA3 (0.53) HSD17B10LMNAALDH1A1AGTR1HIF1A
SCHEMBL9824964 0.82 CACNA1C (0.49) LMNAALDH1A1RAB9AHIF1AMAPT
SCHEMBL10488355 0.81 ADORA3 (0.53) HSD17B10LMNAALDH1A1AGTR1HIF1A
SCHEMBL7406051 0.81 ADORA3 (0.53) HSD17B10LMNAALDH1A1AGTR1HIF1A
SCHEMBL7287257 0.81 ADORA3 (0.53) HSD17B10LMNAALDH1A1AGTR1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276122-A2 Cycloalkyl-substituted 4-aminophenyl halo derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-27 EP disclosed
US-4727082-A CARDIOVASCULAR DISORDERS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1988-02-23 US disclosed
EP-0167371-A2 Dihydropyridine compounds, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1986-01-08 EP disclosed