SCHEMBL9690140

SCHEMBL9690140

CS(=O)(=O)OCCCCCCN1CCN(c2nc(N3CCCC3)nc(N3CCCC3)n2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MMP9 P14780 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
HRH3 Q9Y5N1 4/20 0.39
KMT5A Q9NQR1 8/20 0.38
HTR1A P08908 2/20 0.37
HTR7 P34969 2/20 0.37
TLR9 Q9NR96 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
MAOB P27338 2/20 0.37
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689044 0.90 CASP1 (0.49) MEN1KMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL9690146 0.80 MEN1 (0.59) MEN1KMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL15884868 0.76 ALDH1A1 (0.54) MEN1KMT2ACYP2C19KDM4EUSP2
SCHEMBL6186091 0.74 KDM4E (0.52) KDM4EUSP2ALDH1A1LMNAMMP9
SCHEMBL9689120 0.74 KCNH2 (0.62) ALDH1A1HRH3HTR1AHTR7MAOB
SCHEMBL9689521 0.73 MEN1 (0.72) MEN1KMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL10554729 0.72 KDM4E (0.54) KDM4EUSP2ALDH1A1LMNAMMP9
SCHEMBL24476803 0.72 ALDH1A1 (0.50) MEN1KMT2AKDM4EUSP2ALDH1A1
SCHEMBL5491410 0.72 ALDH1A1 (0.50) MEN1KMT2AKDM4EUSP2ALDH1A1
SCHEMBL9689154 0.71 CASP1 (0.50) KMT5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed