SCHEMBL9691628

SCHEMBL9691628

CCCCOC(=O)OC1=C(C)NC2=C(C(=O)OC2)C1c1ccccc1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
CACNA1F O60840 1/20 0.39
CACNA1D Q01668 1/20 0.39
CACNA1S Q13698 1/20 0.39
CACNA1C Q13936 1/20 0.39
HPGD P15428 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691230 0.97 KDM4E (0.46) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL9690779 0.97 KDM4E (0.46) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL9689489 0.92 KDM4E (0.53) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL9837258 0.89 ALDH1A1 (0.50) KDM4EALDH1A1HPGD
SCHEMBL10817411 0.88 ALDH1A1 (0.51) KDM4EALDH1A1HPGD
SCHEMBL11008926 0.88 KDM4E (0.58) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL9691609 0.87 CACNA1C (0.45) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL9691237 0.87 KDM4E (0.48) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL9691795 0.86 KDM4E (0.45) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL11168071 0.85 KDM4E (0.43) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed
EP-0071819-A1 Dihydropyridines with a positive inotropic activity, their use in pharmaceutical preparations, and processes for their preparation BAYER AG (DE) 1983-02-16 EP disclosed