SCHEMBL9693115

SCHEMBL9693115

COc1cc(Cl)c(CCN2CCC(S(=O)(=O)c3ccc(NS(C)(=O)=O)cc3)CC2)cc1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.48
HTR2A P28223 8/20 0.48
HTR2C P28335 7/20 0.48
DRD2 P14416 4/20 0.48
HTR1A P08908 1/20 0.47
SLC6A4 P31645 1/20 0.47
ABCB1 P08183 1/20 0.42
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
ADRA1D P25100 1/20 0.41
EPHX2 P34913 1/20 0.38
ALDH1A1 P00352 3/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9678100 0.84 KCNH2 (0.48) KCNH2HTR2AHTR2CHTR1ASLC6A4
SCHEMBL9677488 0.71 KCNH2 (0.55) KCNH2HTR2AHTR2CALDH1A1CYP3A4
SCHEMBL9678360 0.71 KCNH2 (0.69) KCNH2HTR2AHTR2CDRD2HTR1A
SCHEMBL9444367 0.70 ABCB1 (0.61) HTR1ASLC6A4ABCB1ALDH1A1LMNA
SCHEMBL6585372 0.69 KCNH2 (0.51) KCNH2HTR2AHTR2CDRD2
SCHEMBL9681410 0.69 ABCB1 (0.43) KCNH2HTR1ASLC6A4ABCB1ALDH1A1
SCHEMBL9447564 0.68 ABCB1 (0.45) KCNH2HTR1ASLC6A4ABCB1ADRA1A
SCHEMBL9041547 0.68 ABCB1 (0.43) KCNH2HTR1ASLC6A4ABCB1ALDH1A1
SCHEMBL7026059 0.68 HTR2A (0.56) KCNH2HTR2AHTR2CDRD2HTR1A
SCHEMBL7022853 0.68 HTR2A (0.52) KCNH2HTR2AHTR2CADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082850-A PIPERIDINE DERIVATIVES AND THERAPEUTIC AND PREVENTIVE AGENTS FOR ARRHYTHMIA CONTAINING SAME EISAI CO., LTD. (JP) 1992-01-21 US disclosed
US-4977165-A Piperidine derivative and therapeutic and preventive agents for arrhythmia containing same EISAI CO., LTD. (JP) 1990-12-11 US disclosed