SCHEMBL9693445

SCHEMBL9693445

O=C(c1ccccc1)N1CCN(c2ccc3nc4[nH]c(=O)[nH]c4cc3c2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 16/20 1.00
PDE3A Q14432 16/20 1.00
C1S P09871 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691872 0.88 PDE3B (0.78) PDE3BPDE3A
SCHEMBL9692111 0.86 PDE3B (1.00) PDE3BPDE3A
SCHEMBL9693701 0.83 PDE3B (1.00) PDE3BPDE3A
SCHEMBL9693383 0.80 PDE3B (1.00) PDE3BPDE3A
SCHEMBL9692011 0.80 PDE3B (1.00) PDE3BPDE3A
SCHEMBL9691765 0.79 PDE3B (1.00) PDE3BPDE3A
SCHEMBL9693319 0.79 PDE3B (1.00) PDE3BPDE3A
SCHEMBL9694200 0.77 PDE3B (0.77) PDE3BPDE3A
SCHEMBL9693683 0.77 PDE3B (1.00) PDE3BPDE3A
SCHEMBL7025618 0.77 PDE3B (0.62) PDE3BPDE3AC1SMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252503-B1 AMINOIMIDAZOQUINOLINE DERIVATIVES Bristol-Myers Squibb Company (US) 1992-11-19 EP claimed
EP-0252503-A1 Aminoimidazoquinoline derivatives Bristol-Myers Squibb Company (US) 1988-01-13 EP claimed
US-4701459-A 7-amino-1,3-dihydro-2H-imidazo[4,5-b]quinolin 2-ones and method for inhibiting phosphodiesterase and blood platelet aggregation BRISTOL-MYERS COMPANY (US) 1987-10-20 US claimed
EP-0252503-B1 AMINOIMIDAZOQUINOLINE DERIVATIVES Bristol-Myers Squibb Company (US) 1992-11-19 EP disclosed
US-4701459-A 7-amino-1,3-dihydro-2H-imidazo[4,5-b]quinolin 2-ones and method for inhibiting phosphodiesterase and blood platelet aggregation BRISTOL-MYERS COMPANY (US) 1987-10-20 US disclosed