SCHEMBL9696134

SCHEMBL9696134

CC(C)c1c(CO)c(-c2ccc(F)cc2)n2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GCGR P47871 13/20 0.39
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
BAZ2B Q9UIF8 1/20 0.36
BAZ2A Q9UIF9 1/20 0.36
FLT3 P36888 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9696278 0.78 IDO1 (0.44) KDM4EMEN1KMT2AALDH1A1GAA
SCHEMBL10335844 0.77 GCGR (0.38) GCGRKDM4EMEN1KMT2AGAA
SCHEMBL9696170 0.76 GCGR (0.44) GCGRKDM4EMEN1KMT2AALDH1A1
SCHEMBL9697139 0.76 ALDH1A1 (0.41) KDM4EMEN1KMT2AALDH1A1GAA
SCHEMBL10691696 0.73 ALDH1A1 (0.36) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL10693357 0.72 HMGCR (0.46) KDM4EALDH1A1
SCHEMBL9753170 0.72 MAPK14 (0.44) GCGR
SCHEMBL10679732 0.68 HMGCR (0.57)
SCHEMBL6241912 0.68 HMGCR (0.57)
SCHEMBL8877962 0.68 HMGCR (0.53) GCGRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124453-A Treatment of corresponding aldehyde with lithium bis(tri-methylsilyl)amide E. R. SQUIBB & SONS, INC. (US) 1992-06-23 US disclosed
EP-0444532-A1 Phosphorus-containing HMG-CoA reductase inhibitors, new intermediates and method E.R. SQUIBB & SONS, INC. (US) 1991-09-04 EP disclosed
US-5025000-A Anticholesterol, antilipemic agents E. R. SQUIBB & SONS, INC. (US) 1991-06-18 US disclosed
US-4751235-A INHIBIT CHOLESTEROL BIOSINTHESIS SANDOZ PHARM. CORP. (US) 1988-06-14 US disclosed
EP-0265640-A2 Azaindole and indolizine derivatives, processes for their production and their use as pharmaceuticals SANDOZ AG (CH) 1988-05-04 EP disclosed