SCHEMBL9699728

SCHEMBL9699728

Cc1cn(-c2cc(C)c(N)c(C#N)c2)cn1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 3/20 0.46
CYP2E1 P05181 1/20 0.38
CYP2A6 P11509 1/20 0.38
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ABL1 P00519 1/20 0.34
BCR P11274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10679905 0.81 KMT2A (0.33) CYP1A2CYP2C9
SCHEMBL1828556 0.79 NR2E1 (0.43) NR2E1CYP2E1CYP2A6CYP1A2CYP3A4
SCHEMBL22199020 0.79 CYP11B2 (0.43) NR2E1CYP2E1CYP2A6CYP1A2CYP3A4
SCHEMBL9699746 0.77 NR2E1 (0.49) NR2E1CYP2E1CYP2A6CYP1A2CYP3A4
SCHEMBL9701824 0.73 NR2E1 (0.46) NR2E1CYP2E1CYP2A6CYP1A2CYP3A4
SCHEMBL10679875 0.73 KDM4E (0.35) CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL9700802 0.73 NR2E1 (0.46) NR2E1CYP2E1CYP2A6CYP1A2CYP3A4
SCHEMBL13530933 0.71 NR2E1 (0.42) NR2E1CYP2E1CYP2A6CYP1A2CYP3A4
SCHEMBL22199045 0.71 USP30 (0.47) NR2E1CYP2E1CYP2A6CYP1A2CYP3A4
SCHEMBL29637047 0.71 KDM4E (0.56) NR2E1CYP2E1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5171851-A Cardiac stimulant DONG-A PHARM. CO., LTD. (KR) 1992-12-15 US disclosed
EP-0510235-A1 Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same DONG-A PHARM. CO., LTD. (KR) 1992-10-28 EP disclosed