SCHEMBL9700191

SCHEMBL9700191

CNCC1COc2c(Cl)cccc2N1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 8/20 0.36
HTR1A P08908 6/20 0.36
HTR2C P28335 6/20 0.36
HTR7 P34969 6/20 0.36
CYP2D6 P10635 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
AQP1 P29972 1/20 0.35
MOGAT2 Q3SYC2 2/20 0.35
HTR1D P28221 5/20 0.35
CA2 P00918 1/20 0.34
HTR2A P28223 2/20 0.33
HTR6 P50406 2/20 0.33
HTR3A P46098 1/20 0.33
HRH1 P35367 1/20 0.33
GAA P10253 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDCD1LG2 Q9BQ51 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700535 0.81 HTR2C (0.38) HTR5AHTR1AHTR2CHTR7HTR1D
SCHEMBL27642723 0.81 CREBBP (0.39) HTR5AHTR1AHTR2CHTR7HTR1D
SCHEMBL9700331 0.81 MTNR1A (0.40) HTR1AHTR2CHTR7CYP2D6SLC6A2
SCHEMBL11854527 0.75 HTR5A (0.43) HTR5AHTR1AHTR2CHTR7HTR1D
SCHEMBL9699375 0.75 GAA (0.50) HTR5AHTR1AHTR2CHTR7HTR1D
SCHEMBL9700527 0.75 GAA (0.50) HTR5AHTR1AHTR2CHTR7SLC6A4
SCHEMBL9700376 0.75 GAA (0.47) HTR5AHTR1AHTR2CHTR7CYP2D6
SCHEMBL9700358 0.72 GAA (0.47) HTR5AHTR1AHTR2CHTR7GAA
SCHEMBL9700466 0.70 HTR2C (0.31) HTR2CHTR2A
SCHEMBL9700468 0.70 GAA (0.44) HTR2CCYP2D6SLC6A2SLC6A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed