SCHEMBL9700358

SCHEMBL9700358

Clc1cccc2c1OCC(CN1CCSCC1)N2

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
CYP2A13 Q16696 1/20 0.40
MAPT P10636 1/20 0.35
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.31
HTR5A P47898 2/20 0.30
HTR1A P08908 1/20 0.30
HTR2C P28335 1/20 0.30
HTR7 P34969 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699375 0.88 GAA (0.50) GAACYP2A13KDM4EALDH1A1SMN1; SMN2
SCHEMBL9700527 0.88 GAA (0.50) GAAKDM4EALDH1A1SMN1; SMN2HTR5A
SCHEMBL9700376 0.85 GAA (0.47) GAAHTR5AHTR1AHTR2CHTR7
SCHEMBL9700468 0.82 GAA (0.44) GAAMAPTHTR2CMEN1KMT2A
SCHEMBL9701579 0.82 GAA (0.44) GAAKDM4EALDH1A1SMN1; SMN2HTR1A
SCHEMBL9700535 0.76 HTR2C (0.38) GAAHTR5AHTR1AHTR2CHTR7
SCHEMBL27642723 0.76 CREBBP (0.39) GAAHTR5AHTR1AHTR2CHTR7
SCHEMBL9700191 0.72 HTR5A (0.36) GAAHTR5AHTR1AHTR2CHTR7
SCHEMBL9699340 0.72 CYP2A13 (0.39) CYP2A13MAPT
SCHEMBL9700277 0.70 GAA (0.47) GAAALDH1A1HTR1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed