SCHEMBL9699340

SCHEMBL9699340

NN1c2cccc(Cl)c2OCC1CN1CCSCC1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 1/20 0.39
NOTUM Q6P988 1/20 0.34
MAPT P10636 1/20 0.32
KDM1A O60341 2/20 0.32
DRD2 P14416 5/20 0.31
DRD4 P21917 4/20 0.31
DRD5 P21918 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701602 0.89 ADRA2A (0.38) NOTUMDRD2DRD4
SCHEMBL9699278 0.89 NOTUM (0.36) NOTUMDRD2DRD4
SCHEMBL9728710 0.85 DRD2 (0.40) NOTUMDRD2DRD4DRD3
SCHEMBL9700270 0.83 CYP2A13 (0.37) CYP2A13NOTUMMAPTDRD2DRD4
SCHEMBL9728617 0.82 ADRA1A (0.41)
SCHEMBL9699323 0.81 CXCR4 (0.36) DRD2DRD3
SCHEMBL9699269 0.79 NOTUM (0.38) NOTUMDRD2
SCHEMBL10378979 0.77 ADRA1A (0.38)
SCHEMBL9700368 0.74 NOTUM (0.37) NOTUM
SCHEMBL9699297 0.72 NOTUM (0.38) NOTUMDRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed