SCHEMBL9700412

SCHEMBL9700412

COc1cc2c3c(c1)c(Sc1ccccc1)c(C)n3C(CN)CO2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.33
DRD3 P35462 2/20 0.33
CNR1 P21554 3/20 0.33
CNR2 P34972 3/20 0.33
MEN1 O00255 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
AKR1B1 P15121 2/20 0.32
PTGDR2 Q9Y5Y4 2/20 0.32
CYP19A1 P11511 2/20 0.32
TUBB4A P04350 2/20 0.32
TUBB P07437 2/20 0.32
TUBA3C P0DPH7 2/20 0.32
TUBA1B P68363 2/20 0.32
TUBA4A P68366 2/20 0.32
TUBB4B P68371 2/20 0.32
TUBB3 Q13509 2/20 0.32
TUBB2A Q13885 2/20 0.32
TUBB8 Q3ZCM7 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700074 0.88 TUBB4A (0.33) DRD2DRD3CNR1CNR2MEN1
SCHEMBL9700330 0.87 CNR1 (0.40) DRD2DRD3CNR1CNR2MEN1
SCHEMBL9701551 0.87 CNR1 (0.40) DRD2DRD3CNR1CNR2MEN1
SCHEMBL9699362 0.86 CNR1 (0.39) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9700286 0.86 PTGDR2 (0.34) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9701364 0.85 CNR1 (0.38) DRD2DRD3CNR1CNR2MEN1
SCHEMBL9700401 0.82 CNR1 (0.36) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9700394 0.81 TUBB4A (0.30) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL9701576 0.74 PTGDR2 (0.33) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9699279 0.74 CNR1 (0.45) CNR1CNR2MEN1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed