SCHEMBL9700598

SCHEMBL9700598

CS(=O)(=O)N1CC(CN2CCOCC2)Oc2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
SCN1A P35498 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN3A Q9NY46 1/20 0.42
DRD2 P14416 3/20 0.40
ABCB1 P08183 1/20 0.40
HTR2A P28223 1/20 0.40
HRH1 P35367 1/20 0.40
GAA P10253 1/20 0.39
HTR1A P08908 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
HTR7 P34969 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700324 0.80 ADRA2A (0.47) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL10379007 0.79 POLB (0.43) GAAALDH1A1CA2
SCHEMBL9700502 0.78 ADRA2A (0.45) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9455117 0.75 CASR (0.45) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL5582588 0.75 RORC (0.42) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL20090898 0.72 MEN1 (0.40) ABCB1GAAHTR1ASIGMAR1ALDH1A1
SCHEMBL9699315 0.72 CNR1 (0.47) GAAALDH1A1
SCHEMBL9699068 0.71 LMNA (0.43) GAAALDH1A1
SCHEMBL5582757 0.71 RORC (0.42) GAAALDH1A1
SCHEMBL9699072 0.70 LMNA (0.44) GAAALDH1A1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed