SCHEMBL9700631

SCHEMBL9700631

COc1cc2nc(CBr)c(CBr)nc2cc1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.52
PGK1 P00558 8/20 0.50
ALDH1A1 P00352 4/20 0.41
PDGFRB P09619 2/20 0.41
PDGFRA P16234 2/20 0.41
RPS6KB2 Q9UBS0 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 2/20 0.40
GLA P06280 2/20 0.40
GAA P10253 2/20 0.40
MAPT P10636 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ERBB2 P04626 1/20 0.40
GSK3B P49841 1/20 0.40
MAP4K2 Q12851 1/20 0.40
HPGD P15428 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11487596 0.88 NQO2 (0.46) NQO2PGK1ALDH1A1PDGFRBPDGFRA
SCHEMBL11477391 0.88 NQO2 (0.46) NQO2PGK1ALDH1A1PDGFRBPDGFRA
SCHEMBL9701973 0.83 NQO2 (0.39) NQO2PGK1ALDH1A1KDM4EGLA
SCHEMBL11696562 0.80 PDE4A (0.54) NQO2PGK1ALDH1A1PDGFRBPDGFRA
SCHEMBL30932234 0.76 ALDH1A1 (0.61) NQO2ALDH1A1PDGFRBPDGFRASMN1; SMN2
SCHEMBL29600727 0.75 ALDH1A1 (0.40) NQO2PGK1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL571871 0.75 ALDH1A1 (0.40) NQO2PGK1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL1291852 0.75 PGK1 (0.61) NQO2PGK1ALDH1A1PDGFRBPDGFRA
SCHEMBL4177978 0.75 ERBB2 (0.61) NQO2ALDH1A1PDGFRBSMN1; SMN2KDM4E
SCHEMBL29029328 0.74 NQO2 (0.62) NQO2PGK1ALDH1A1PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992014740-A1 QUINOXALINE PHOSPHONO-AMINO ACIDS AMERICAN HOME PRODUCTS CORPORATION (US) 1992-09-03 WO disclosed
US-5118675-A Therapy for central nervous system disorders AMERICAN HOME PRODUCTS CORPORATION (US) 1992-06-02 US disclosed