SCHEMBL9701973

SCHEMBL9701973

COc1cc2nc(CBr)c(CP(=O)(O)O)nc2cc1OC

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.39
PGK1 P00558 4/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
ENPP1 P22413 2/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700631 0.83 NQO2 (0.52) NQO2PGK1KDM4EALDH1A1GLA
SCHEMBL9700929 0.80 GGPS1 (0.39) PGK1
SCHEMBL9702005 0.77
SCHEMBL11487596 0.74 NQO2 (0.46) NQO2PGK1KDM4EALDH1A1GLA
SCHEMBL11477391 0.74 NQO2 (0.46) NQO2PGK1KDM4EALDH1A1GLA
SCHEMBL9746062 0.72 MMP1 (0.36)
SCHEMBL9701697 0.71 ERBB2 (0.44) NQO2KDM4EMAPT
SCHEMBL11696562 0.70 PDE4A (0.54) NQO2PGK1KDM4EALDH1A1GLA
SCHEMBL9699664 0.70 MMP1 (0.41) NQO2PGK1ALDH1A1
SCHEMBL15949820 0.69 STING1 (0.49) ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992014740-A1 QUINOXALINE PHOSPHONO-AMINO ACIDS AMERICAN HOME PRODUCTS CORPORATION (US) 1992-09-03 WO disclosed
US-5118675-A Therapy for central nervous system disorders AMERICAN HOME PRODUCTS CORPORATION (US) 1992-06-02 US disclosed