SCHEMBL9701085

SCHEMBL9701085

CC(C)CCN1Cc2cccc(N)c2NCC1(C)C

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
TLR9 Q9NR96 1/20 0.33
VDR P11473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701190 0.77 SIGMAR1 (0.33)
SCHEMBL9700201 0.66 DRD1 (0.33)
SCHEMBL3587267 0.62 BRD4 (0.54) KEAP1NFE2L2
SCHEMBL12714314 0.61 PARP1 (0.50) KEAP1NFE2L2TLR9VDR
SCHEMBL7902262 0.60 HTR1A (0.39)
SCHEMBL7652793 0.60 MAOA (0.37)
SCHEMBL25080719 0.58 NAMPT (0.57)
SCHEMBL3596149 0.57 PARP1 (0.49)
SCHEMBL3593434 0.57 PARP1 (0.47)
SCHEMBL1119383 0.56 CD44 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992013860-A1 NEW 4,5,6,7-TETRAHYDRO-IMIDAZO-[4,5,lJK][1,4]-BENZODIAZEPINE-2-(1H)-THIONES, A METHOD OF PREPARING THEM AS WELL AS DRUGS CONTAINING THEM, AND INTERMEDIATES FOR THE PREPARATION OF THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1992-08-20 WO disclosed