SCHEMBL9701383

SCHEMBL9701383

COc1cccc2c1OCC(CN1CCCC1)N2

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
POLB P06746 1/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
KMT2A Q03164 1/20 0.39
HRH3 Q9Y5N1 5/20 0.38
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
CHRNA7 P36544 1/20 0.37
HTR1A P08908 1/20 0.36
KDM2B Q8NHM5 1/20 0.36
KCNH2 Q12809 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700277 0.97 GAA (0.47) GAAPOLBMEN1ALDH1A1CYP1A2
SCHEMBL9701643 0.91 GAA (0.42) GAACYP1A2CYP2D6HTR1A
SCHEMBL9700342 0.90 GAA (0.45) GAAHRH3ADRA2AADRA2BADRA2C
SCHEMBL9701579 0.89 GAA (0.44) GAAMEN1ALDH1A1KMT2AADRA2A
SCHEMBL9700527 0.81 GAA (0.50) GAAPOLBMEN1ALDH1A1KMT2A
SCHEMBL9701412 0.80 HTR1A (0.40) GAAALDH1A1HTR1A
SCHEMBL9699375 0.78 GAA (0.50) GAAPOLBMEN1ALDH1A1KMT2A
SCHEMBL9700331 0.78 MTNR1A (0.40) GAAMEN1ALDH1A1CYP1A2CYP2D6
SCHEMBL9701616 0.73 GAA (0.77) GAAALDH1A1ADRA2AADRA2BADRA2C
SCHEMBL9701640 0.73 CHRNB4 (0.38) CYP2D6ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed