SCHEMBL9701643

SCHEMBL9701643

COc1cccc2c1OCC(CN1CCCNCC1)N2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
HTR7 P34969 2/20 0.36
HTR1A P08908 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
ADRB1 P08588 1/20 0.35
DRD2 P14416 1/20 0.35
CYP2C19 P33261 1/20 0.35
DRD3 P35462 1/20 0.35
HTR3A P46098 1/20 0.35
HTR6 P50406 1/20 0.35
HTR3D Q70Z44 1/20 0.35
HTR3C Q8WXA8 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
CXCR4 P61073 1/20 0.35
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700277 0.91 GAA (0.47) GAAHTR1AADRA1AADRA1BCYP1A2
SCHEMBL9701383 0.91 GAA (0.47) GAAHTR1ACYP1A2CYP2D6
SCHEMBL9700342 0.84 GAA (0.45) GAAHTR1AADRA1ADRD2DRD3
SCHEMBL9700468 0.83 GAA (0.44) GAAADRB1DRD2DRD3SIGMAR1
SCHEMBL9701579 0.83 GAA (0.44) GAAHTR7HTR1AADRA1DADRA1A
SCHEMBL9699287 0.77 HTR7 (0.40) HTR7HTR1AADRA1DADRA1AADRA1B
SCHEMBL9701412 0.75 HTR1A (0.40) GAAHTR7HTR1AADRA1DADRA1A
SCHEMBL9701640 0.75 CHRNB4 (0.38) ADRA1DADRA1AADRA1BSLC6A4CYP2D6
SCHEMBL9701648 0.74 LMNA (0.41) HTR7HTR1AADRA1DADRA1AADRA1B
SCHEMBL9699375 0.73 GAA (0.50) GAAHTR7HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed